SCHEMBL8936909

SCHEMBL8936909

CC(c1ccccc1OCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)N(C)CCC1(OC(=O)C(=O)OC2(CCN(C)C(C)c3ccccc3OCc3cc(C(F)(F)F)cc(C(F)(F)F)c3)N=NN=N2)N=NN=N1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 13/20 0.38
GPBAR1 Q8TDU6 1/20 0.36
SLC1A5 Q15758 1/20 0.36
MME P08473 1/20 0.35
ACE P12821 1/20 0.35
CPA1 P15085 1/20 0.35
ACE2 Q9BYF1 1/20 0.35
KIFC1 Q9BW19 1/20 0.35
CCR2 P41597 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.34
PTPN1 P18031 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936903 0.92 TACR1 (0.39) TACR1GPBAR1SLC1A5MMEACE
SCHEMBL8936931 0.73 TACR1 (0.40) TACR1
SCHEMBL8936871 0.73 TACR1 (0.45) TACR1
SCHEMBL8936863 0.71 TACR1 (0.45) TACR1
SCHEMBL8936826 0.70 TACR1 (0.61) TACR1
SCHEMBL8936832 0.70 TACR1 (0.61) TACR1
SCHEMBL8936828 0.66 TACR1 (0.38) TACR1PTPN1
SCHEMBL8936907 0.66 TACR1 (0.64) TACR1
SCHEMBL8936904 0.66 TACR1 (0.63) TACR1
SCHEMBL5793298 0.65 MAPT (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5494926-A ANTIINFLAMMATORY AGENT, ANTIARTHRITIC AGENT; TREATING PAIN, HEADACHE MERCK SHARP & DOHME LTD. (GB) 1996-02-27 US disclosed