SCHEMBL8938264

SCHEMBL8938264

CCOC(=O)c1cc2cc(Cl)ccc2n1S(=O)(=O)c1ccccc1.Cc1cccc(S(N)(=O)=O)c1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOD2 Q9HC29 4/20 0.64
NOD1 Q9Y239 4/20 0.64
PPARG P37231 9/20 0.54
PPARA Q07869 7/20 0.54
PPARD Q03181 5/20 0.54
BCL2 P10415 1/20 0.42
BID P55957 1/20 0.42
MCL1 Q07820 1/20 0.42
ELANE P08246 1/20 0.41
CHRNA7 P36544 1/20 0.41
ACLY P53396 2/20 0.40
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzenesulfonamide SCHEMBL8938299 0.93 NOD2 (0.70) NOD2NOD1PPARGPPARAPPARD
SCHEMBL2347003 0.90 NOD2 (0.78) NOD2NOD1PPARGPPARAPPARD
SCHEMBL8938381 0.85 NOD2 (0.64) NOD2NOD1PPARGPPARAPPARD
SCHEMBL22003860 0.81 NOD2 (0.69) NOD2NOD1PPARGPPARAPPARD
SCHEMBL16486105 0.79 NOD2 (0.58) NOD2NOD1PPARGPPARAPPARD
SCHEMBL3141535 0.79 NOD2 (0.69) NOD2NOD1PPARGPPARAPPARD
SCHEMBL2542152 0.78 NOD2 (0.86) NOD2NOD1BCL2BIDMCL1
SCHEMBL10003942 0.78 NOD2 (0.78) NOD2NOD1PPARGPPARAPPARD
SCHEMBL13114472 0.76 NOD2 (0.81) NOD2NOD1PPARGPPARDBCL2
SCHEMBL3837213 0.75 PPARG (0.61) NOD2NOD1PPARGPPARAPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527819-A TREATING AIDS MERCK & CO., INC. (US) 1996-06-18 US disclosed
EP-0686148-A4 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO INC (US) 1996-02-07 EP disclosed
EP-0686148-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO. INC. (US) 1995-12-13 EP disclosed
WO-1994019321-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1994-09-01 WO disclosed