SCHEMBL8938522

SCHEMBL8938522

O=C(NCc1cccnc1)c1[nH]c2ccc(Cl)cc2c1S(=O)(=O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 12/20 0.55
NPSR1 Q6W5P4 2/20 0.49
LMNA P02545 2/20 0.49
HTT P42858 2/20 0.49
GAA P10253 1/20 0.48
CYP2C9 P11712 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
PKM P14618 1/20 0.48
HPGD P15428 1/20 0.48
CYP2C19 P33261 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
ALDH1A1 P00352 1/20 0.47
TUBB4A P04350 1/20 0.46
TUBB P07437 1/20 0.46
TUBA3C P0DPH7 1/20 0.46
TUBA1B P68363 1/20 0.46
TUBA4A P68366 1/20 0.46
TUBB4B P68371 1/20 0.46
TUBB3 Q13509 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8938481 0.90 TUBB (0.53) ALDH1A1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8938242 0.85 TUBB4A (0.46) NAMPTNPSR1ALDH1A1TUBB4ATUBB
SCHEMBL8938465 0.85 TUBB (0.50) ALDH1A1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8938426 0.85 TUBB (0.49) NAMPTALDH1A1TUBB4ATUBBTUBA3C
SCHEMBL8938397 0.84 TUBB4A (0.49) NAMPTALDH1A1TUBB4ATUBBTUBA3C
SCHEMBL8938394 0.84 TUBB4A (0.45) NAMPTNPSR1CYP2C9ALDH1A1TUBB4A
SCHEMBL8938410 0.83 HPGD (0.51) LMNAHTTHPGDALDH1A1TUBB4A
SCHEMBL9034050 0.82 CNR1 (0.66) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL8938246 0.82 CNR1 (0.58) NAMPTTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8938452 0.82 TUBB4A (0.66) LMNATUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686148-A4 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO INC (US) 1996-02-07 EP claimed
EP-0686148-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO. INC. (US) 1995-12-13 EP claimed
WO-1994019321-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1994-09-01 WO claimed
US-5527819-A TREATING AIDS MERCK & CO., INC. (US) 1996-06-18 US disclosed
EP-0686148-A4 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO INC (US) 1996-02-07 EP disclosed
EP-0686148-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO. INC. (US) 1995-12-13 EP disclosed
WO-1994019321-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1994-09-01 WO disclosed