SCHEMBL8938557

SCHEMBL8938557

O=C(NCCCn1ccnc1)c1[nH]c2ccc(Cl)cc2c1S(=O)(=O)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.53
MEN1 O00255 1/20 0.53
ALDH1A1 P00352 2/20 0.52
KDM4E B2RXH2 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
CDK1 P06493 1/20 0.48
CDK2 P24941 1/20 0.48
NAMPT P43490 1/20 0.48
LMNA P02545 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8938246 0.81 CNR1 (0.58) NAMPT
SCHEMBL8938285 0.80 CNR1 (0.49)
SCHEMBL9034050 0.79 CNR1 (0.66) CDK2
SCHEMBL9033484 0.79 NAMPT (0.46) NAMPT
SCHEMBL8938277 0.78 TUBB4A (0.47) ALDH1A1KDM4ECDK2NAMPTMAPT
SCHEMBL8938345 0.78 CNR1 (0.49) CDK2
SCHEMBL8938511 0.78 TUBB4A (0.56) ALDH1A1KDM4EMAPT
SCHEMBL8938368 0.78 TUBB4A (0.47) ALDH1A1KDM4ENAMPTLMNASMN1; SMN2
SCHEMBL8938466 0.77 CNR1 (0.49) ALDH1A1KDM4E
SCHEMBL8938481 0.77 TUBB (0.53) KMT2AMEN1ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527819-A TREATING AIDS MERCK & CO., INC. (US) 1996-06-18 US disclosed
WO-1994019321-A1 INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1994-09-01 WO disclosed