SCHEMBL8939156

SCHEMBL8939156

Cc1ccc(CN2CCC(Oc3cc4cc[nH]c(=O)c4cc3C)CC2)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 4/20 0.52
MAP2K1 Q02750 2/20 0.46
OPRM1 P35372 5/20 0.46
OPRD1 P41143 3/20 0.46
OPRK1 P41145 3/20 0.46
CACNA1F O60840 2/20 0.46
CHRM1 P11229 2/20 0.46
ADRA1D P25100 2/20 0.46
HTR7 P34969 2/20 0.46
ADRA1A P35348 2/20 0.46
ADRA1B P35368 2/20 0.46
OPRL1 P41146 2/20 0.46
CACNA1D Q01668 2/20 0.46
CACNA1S Q13698 2/20 0.46
CACNA1C Q13936 2/20 0.46
CHRM2 P08172 1/20 0.46
DRD2 P14416 1/20 0.46
DRD1 P21728 1/20 0.46
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8938694 0.94 MAP2K1 (0.54) ROCK1MAP2K1OPRM1OPRD1OPRK1
SCHEMBL8937948 0.93 ROCK1 (0.52) ROCK1MAP2K1OPRM1HRH1CCR3
SCHEMBL8937951 0.90 ROCK1 (0.52) ROCK1MAP2K1OPRM1DRD4MEN1
SCHEMBL8937943 0.88 ROCK1 (0.56) ROCK1MAP2K1OPRM1ROCK2PRKACA
SCHEMBL8938636 0.86 ROCK1 (0.53) ROCK1OPRM1OPRD1OPRK1CACNA1F
SCHEMBL8938824 0.86 OPRM1 (0.48) ROCK1OPRM1OPRD1OPRK1CACNA1F
SCHEMBL8937994 0.85 ROCK1 (0.55) ROCK1MAP2K1OPRM1DRD2DRD4
SCHEMBL8934976 0.84 MAP2K1 (0.56) ROCK1MAP2K1OPRM1ROCK2MEN1
SCHEMBL8937925 0.84 ROCK1 (0.54) ROCK1MAP2K1ROCK2PRKACAPRKCD
SCHEMBL8937945 0.84 ROCK1 (0.56) ROCK1MAP2K1ROCK2PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed