6-[(Isopropyl)Oxy]Purine

6-[(Isopropyl)Oxy]Purine

SCHEMBL8939256

CC(C)Oc1ncnc2[nH]cnc12

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 3/20 0.44
CDK1 P06493 3/20 0.44
CCNB1 P14635 2/20 0.44
CCNA2 P20248 2/20 0.44
CCNA1 P78396 2/20 0.44
MAP3K7 O43318 9/20 0.42
TAB1 Q15750 9/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PDPK1 O15530 1/20 0.36
TTBK1 Q5TCY1 1/20 0.35
TTBK2 Q6IQ55 1/20 0.35
LRRK2 Q5S007 1/20 0.34
MAP4K4 O95819 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL284829 0.79 PDPK1 (0.52) PDPK1TTBK1TTBK2
SCHEMBL12270784 0.79 MAP3K7 (0.50) CDK2CDK1CCNB1CCNA2CCNA1
SCHEMBL9682496 0.78 CDK2 (0.59) CDK2CDK1CCNB1CCNA2CCNA1
SCHEMBL2940695 0.77 PDPK1 (0.36) PDPK1LRRK2
SCHEMBL3388862 0.76 KDM4E (0.40) CDK2CDK1CCNB1CCNA2CCNA1
SCHEMBL2623129 0.76 CDK1 (0.50) CDK2CDK1CCNB1CCNA2CCNA1
SCHEMBL16549309 0.75 CDK2 (0.41) CDK2CDK1CCNB1CCNA2CCNA1
SCHEMBL17924977 0.72 PDPK1 (0.34) PDPK1
SCHEMBL22639807 0.72 CDK1 (0.48) CDK2CDK1CCNB1CCNA2CCNA1
SCHEMBL2938606 0.72 MAP3K7 (0.37) MAP3K7TAB1KDM4EPDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5574149-A Method of treating HIV infections with 2',3'-dideoxy-3'-fluoro-5-chlorouridine GLAXO WELLCOME INC. (US) 1996-11-12 US disclosed
EP-0586523-A4 DETERMINATION OF PRODRUGS METABOLIZABLE BY THE LIVER AND THERAPEUTIC USE THEREOF UNIV YALE (US) 1995-11-29 EP disclosed
EP-0670328-A1 Therapeutic nucleosides THE WELLCOME FOUNDATION LIMITED (GB) 1995-09-06 EP disclosed
EP-0669341-A1 Therapeutic Nucleosides THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-30 EP disclosed
EP-0586523-A1 DETERMINATION OF PRODRUGS METABOLIZABLE BY THE LIVER AND THERAPEUTIC USE THEREOF YALE UNIVERSITY (US) 1994-03-16 EP disclosed
US-5213972-A Production of thymidine and deoxyuridine, intermediates for AZT CHEMGEN CORPORATION (US) 1993-05-25 US disclosed
EP-0317128-A2 Anti-HIV Pyrimidine Nucleosides THE WELLCOME FOUNDATION LIMITED (GB) 1989-05-24 EP disclosed