SCHEMBL8941781

SCHEMBL8941781

CC1Cc2ccccc2-c2ccccc21

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.59
HTR2A P28223 2/20 0.53
NOTUM Q6P988 2/20 0.46
NOS3 P29474 2/20 0.44
NOS2 P35228 2/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
CYP19A1 P11511 2/20 0.41
CYP11B2 P19099 2/20 0.41
NOS1 P29475 1/20 0.40
GPR3 P46089 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
TYMS P04818 1/20 0.40
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
CDK8 P49336 1/20 0.39
CDK5 Q00535 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14555189 0.81 HTR2A (0.50) ACHEHTR2ANOS3NOS2NOS1
SCHEMBL31554961 0.81
SCHEMBL371454 0.81
SCHEMBL19388157 0.81
SCHEMBL14770098 0.80 ACHE (0.47) ACHEHTR2ANOTUMNOS3NOS2
SCHEMBL22933878 0.80 ACHE (0.43) ACHEHTR2ANOTUMNOS3NOS2
Ammonia Solution, Strong SCHEMBL11220000 0.79 HTR2A (0.48) ACHEHTR2ANOS3NOS2NOS1
SCHEMBL1200699 0.77 ACHE (0.56) ACHEHTR2ANOS3NOS2TSHR
SCHEMBL14169777 0.76 HTR2A (0.47) ACHEHTR2ANOTUMNOS3NOS2
SCHEMBL29439854 0.76 HTR2A (0.55) ACHEHTR2ANOS3NOS2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5480913-A DIHYDRO-PHENANTHRENE DERIVATIVES, SIDE EFFECT REDUCTION ARCH DEVELOPMENT CORPORATION (US) 1996-01-02 US disclosed
EP-0363128-B1 ANTI-ANDROGEN COMPOUNDS ARCH DEVELOPMENT CORPORATION (US) 1993-09-01 EP disclosed
US-5208263-A Dihydrophenanthrene derivatives ARCH DEVELOPMENT CORPORATION (US) 1993-05-04 US disclosed
WO-1990003979-A2 ANTI-ANDROGEN COMPOUNDS ARCH DEVELOPMENT CORPORATION (US) 1990-04-19 WO disclosed
EP-0363128-A2 Anti-androgen compounds ARCH DEVELOPMENT CORPORATION (US) 1990-04-11 EP disclosed