SCHEMBL8941949

SCHEMBL8941949

CCNC1CN(c2cc3nc4c(cc3cc2F)c(=O)c(C(=O)O)cn4NC)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 2/20 0.39
LMNA P02545 5/20 0.38
CYP2C9 P11712 1/20 0.38
ATP6V1B2 P21281 1/20 0.38
TBXA2R P21731 1/20 0.38
EDNRA P25101 1/20 0.38
TARBP2 Q15633 1/20 0.38
KDM4E B2RXH2 8/20 0.38
ALDH1A1 P00352 7/20 0.38
HPGD P15428 5/20 0.38
HSD17B10 Q99714 5/20 0.38
HTT P42858 3/20 0.38
POLB P06746 1/20 0.38
XBP1 P17861 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
DRD3 P35462 1/20 0.38
MAPT P10636 1/20 0.38
EPHA2 P29317 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8941940 0.91 ALDH1A1 (0.39) TOP1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8942035 0.91 TOP1 (0.38) TOP1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8942041 0.91 TOP1 (0.42) TOP1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8942032 0.89 DRD3 (0.41) TOP1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8942236 0.89 TOP1 (0.39) TOP1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8941913 0.89 LMNA (0.51) TOP1LMNACYP2C9ATP6V1B2TBXA2R
Water SCHEMBL8942061 0.89 DRD3 (0.40) TOP1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8942031 0.87 KMT2A (0.46) TOP1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8942103 0.87 LMNA (0.38) TOP1LMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8942126 0.87 KDM4E (0.49) TOP1LMNACYP2C9KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556861-A 1,8 benzonaphthyridine derivatives and antimicrobial compositions LABORATOIRE ROGER BELLON (FR) 1996-09-17 US disclosed