SCHEMBL8942258

SCHEMBL8942258

C=C1N(CCOC(C)=O)c2ccccc2C1(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.47
OPRK1 P41145 1/20 0.47
OPRL1 P41146 1/20 0.47
SLC18A3 Q16572 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 7/20 0.39
ALDH1A1 P00352 5/20 0.39
PKM P14618 1/20 0.39
LMNA P02545 4/20 0.38
TP53 P04637 3/20 0.38
THRB P10828 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
NPC1 O15118 1/20 0.37
ALPL P05186 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9222528 0.88 OPRM1 (0.38) OPRM1OPRK1OPRL1CYP1A2CYP2D6
SCHEMBL4982011 0.81 KMT2A (0.44) CYP1A2CYP2D6KMT2AMAPTALDH1A1
SCHEMBL9089556 0.79 POLB (0.42) OPRL1CYP1A2CYP2D6KMT2ALMNA
SCHEMBL10883795 0.79 SMN1; SMN2 (0.46) OPRM1OPRK1OPRL1KMT2AMAPT
SCHEMBL19116479 0.79 KMT2A (0.42) OPRL1CYP1A2CYP2D6KMT2AMAPT
SCHEMBL2180470 0.78 KMT2A (0.46) OPRM1OPRL1CYP1A2CYP2D6KMT2A
SCHEMBL13247890 0.78 KMT2A (0.41) CYP1A2CYP2D6KMT2AMAPTALDH1A1
SCHEMBL14440502 0.78 KMT2A (0.41) OPRL1CYP1A2CYP2D6KMT2AMAPT
SCHEMBL12410885 0.78 KMT2A (0.38) OPRM1OPRK1OPRL1CYP1A2CYP2D6
SCHEMBL14428040 0.77 KMT2A (0.40) CYP1A2CYP2D6KMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578711-A Process for the preparation of dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1996-11-26 US disclosed
US-5541299-A Process for the preparation of dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1996-07-30 US disclosed
US-5502171-A Process for the preparation of dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1996-03-26 US disclosed
EP-0446731-B1 Process for the manufacture of azo dyes BAYER AG (DE) 1995-05-03 EP disclosed
EP-0446731-A2 Process for the manufacture of azo dyes BAYER AG (DE) 1991-09-18 EP disclosed
EP-0087706-B1 CATIONIC HYDRAZONE DYES, THEIR MANUFACTURE AND THEIR USE BAYER AG (DE) 1986-07-30 EP disclosed
US-4496719-A 3H-Indol-2-yl cationic hydrazone dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1985-01-29 US disclosed
EP-0087706-A2 Cationic hydrazone dyes, their manufacture and their use BAYER AG (DE) 1983-09-07 EP disclosed