SCHEMBL8943879

SCHEMBL8943879

Cc1c(F)c(F)c(F)c2c(=O)c(C(=O)O)c(F)n(C3CC3)c12

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 3/20 0.38
TOP2B Q02880 3/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
STAT3 P40763 1/20 0.33
NOTUM Q6P988 1/20 0.33
KCNH2 Q12809 2/20 0.32
HRH3 Q9Y5N1 1/20 0.32
CACNA1F O60840 1/20 0.32
POLB P06746 1/20 0.32
MAPK1 P28482 1/20 0.32
CACNA1D Q01668 1/20 0.32
CACNA1S Q13698 1/20 0.32
CACNA1C Q13936 1/20 0.32
GSK3B P49841 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.30
TAS1R1 Q7RTX1 1/20 0.30
TAS1R2 Q8TE23 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27520234 0.80 NOTUM (0.37) TOP2ATOP2BMEN1KMT2ANOTUM
SCHEMBL6786216 0.78 GSK3B (0.40) TOP2ATOP2BKCNH2CACNA1FPOLB
SCHEMBL5001847 0.78 TOP2A (0.38) TOP2ATOP2BMEN1KMT2ANOTUM
SCHEMBL8120234 0.75 MEN1 (0.36) TOP2ATOP2BMEN1KMT2ASTAT3
SCHEMBL27408658 0.72 ALDH1A1 (0.41) TOP2ATOP2BMEN1KMT2AKCNH2
SCHEMBL27351360 0.72 MEN1 (0.53) MEN1KMT2AKCNH2HRH3CACNA1F
SCHEMBL27322864 0.70 MEN1 (0.36) TOP2ATOP2BMEN1KMT2ASTAT3
SCHEMBL27610949 0.69 STAT3 (0.36) TOP2ATOP2BMEN1KMT2ASTAT3
SCHEMBL28069524 0.69 TPMT (0.36) MEN1KMT2AKCNH2POLBGSK3B
SCHEMBL15598878 0.68 CACNA1F (0.35) TOP2ATOP2BKCNH2CACNA1FPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5493048-A REACTING METALLIZED FLUORO-TRIFLUOROMETHYLBENZENE DERIVATIVE WITH CARBON DIOXIDE AND PRODUCT IS THEN HYDROLYSED WITH AN ACID TO FORM ACID, SIMILARLY HALOGENATION GIVE ACID HALIDE AND WITH ALCOHOL GIVES ESTER BAYER AKTIENGESELLSCHAFT (DE) 1996-02-20 US disclosed