SCHEMBL8946093

SCHEMBL8946093

CN1C=Nc2ccccc2CC1c1cccs1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
NOS3 P29474 1/20 0.38
NOS2 P35228 1/20 0.38
KDM4E B2RXH2 4/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
PKM P14618 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
POLB P06746 1/20 0.36
ALDH1A1 P00352 5/20 0.36
LMNA P02545 2/20 0.36
HTT P42858 2/20 0.36
HPGD P15428 1/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36
GLA P06280 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11154268 0.78 NPC1 (0.41) SLC6A2SLC6A4SLC6A3SMN1; SMN2ALDH1A1
SCHEMBL8945774 0.77 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3NOS3NOS2
Hydrochloric Acid SCHEMBL9581759 0.77 NPC1 (0.44) SLC6A2SLC6A4SLC6A3KDM4ESMN1; SMN2
SCHEMBL8946091 0.74 SLC6A2 (0.38) SLC6A2SLC6A4SLC6A3NOS3NOS2
SCHEMBL8945788 0.74 MEN1 (0.38) SLC6A2SLC6A4SLC6A3NOS3NOS2
Hydrochloric Acid SCHEMBL8946092 0.73 MEN1 (0.37) SLC6A2SLC6A4SLC6A3NOS3NOS2
Hydrochloric Acid SCHEMBL8945737 0.73 SLC6A2 (0.37) SLC6A2SLC6A4SLC6A3NOS3NOS2
SCHEMBL8945770 0.72 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3NOS3NOS2
Hydrochloric Acid SCHEMBL8945853 0.71 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3NOS3NOS2
SCHEMBL8945814 0.69 GAA (0.44) KDM4EMEN1KMT2AL3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed