SCHEMBL8946193

SCHEMBL8946193

CCOC(=O)CN(c1ccncc1F)n1ccc2cc(OCc3ccccc3)ccc21

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.46
MEN1 O00255 1/20 0.41
HSP90AA1 P07900 1/20 0.41
KMT2A Q03164 1/20 0.41
SRD5A2 P31213 1/20 0.40
MAOB P27338 2/20 0.40
MMP13 P45452 2/20 0.39
NMT1 P30419 2/20 0.39
ROCK1 Q13464 1/20 0.39
PPARG P37231 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946054 0.90 MEN1 (0.41) MEN1HSP90AA1KMT2ASRD5A2MAOB
SCHEMBL8946223 0.88 MEN1 (0.44) BCHEMEN1HSP90AA1KMT2ASRD5A2
SCHEMBL7621050 0.86 BCHE (0.51) BCHEMEN1KMT2ASRD5A2ROCK1
Hydrochloric Acid SCHEMBL8544417 0.85 BCHE (0.51) BCHEMEN1KMT2ASRD5A2ROCK1
SCHEMBL8946048 0.84 BCHE (0.44) BCHEMEN1KMT2ASRD5A2ROCK1
SCHEMBL8946085 0.84 SLC6A2 (0.47) BCHEMEN1KMT2AALDH1A1
SCHEMBL9674458 0.76 ROCK1 (0.46) MEN1KMT2ASRD5A2ROCK1
SCHEMBL8946151 0.74 MEN1 (0.47) BCHEMEN1HSP90AA1KMT2ASRD5A2
SCHEMBL8946189 0.74 ROCK1 (0.43) MEN1KMT2ASRD5A2ROCK1
SCHEMBL8539041 0.73 SLC6A2 (0.71) MEN1KMT2ASRD5A2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0509400-B1 1-(Pyrido[3,4-b]-1,4-oxazinyl-4-yl)-1H-indoles, intermediates and a process for their preparation, and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1996-07-03 EP disclosed
US-5519131-A CYCLIZATION OF HYDROXYALKYLAMINO COMPOUND IN THE PRESENCE OF STRONG BASE SUCH AS SODIUM HYDRIDE OR POTASSIUM TERT-BUTOXIDE HOECHST MARION ROUSSEL INC. (US) 1996-05-21 US disclosed
US-5276156-A Antidepressants, treatment of Alzheimer*s disease HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-01-04 US disclosed
US-5214038-A Cholinesterase inhibitors, antidepressants, cognition activators HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-05-25 US disclosed
EP-0509400-A1 1-(Pyrido[3,4-b]-1,4-oxazinyl-4-yl)-1H-indoles, intermediates and a process for their preparation, and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-10-21 EP disclosed