SCHEMBL8946189

SCHEMBL8946189

OCCN(c1ccncc1Cl)n1ccc2cc(OCc3ccccc3)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.43
SLC6A2 P23975 3/20 0.40
MRGPRX4 Q96LA9 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
SRD5A2 P31213 1/20 0.37
ALOX5 P09917 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
CYP3A4 P08684 2/20 0.35
CYP26A1 O43174 1/20 0.35
GRM2 Q14416 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
EPHB3 P54753 1/20 0.35
LTB4R Q15722 1/20 0.35
LTB4R2 Q9NPC1 1/20 0.35
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946048 0.89 BCHE (0.44) ROCK1SLC6A2MRGPRX4MEN1NPC1
SCHEMBL8946054 0.84 MEN1 (0.41) ROCK1MEN1KMT2ASRD5A2
SCHEMBL7621050 0.80 BCHE (0.51) ROCK1SLC6A2MEN1NPC1RAB9A
Hydrochloric Acid SCHEMBL8544417 0.79 BCHE (0.51) ROCK1SLC6A2MEN1NPC1RAB9A
SCHEMBL9674458 0.76 ROCK1 (0.46) ROCK1SLC6A2MRGPRX4MEN1NPC1
SCHEMBL8539041 0.75 SLC6A2 (0.71) ROCK1SLC6A2MEN1NPC1RAB9A
SCHEMBL8946193 0.74 BCHE (0.46) ROCK1MEN1KMT2ASRD5A2
SCHEMBL8946151 0.73 MEN1 (0.47) ROCK1SLC6A2MRGPRX4MEN1NPC1
SCHEMBL8946215 0.73 SLC6A2 (0.56) ROCK1SLC6A2
SCHEMBL9738604 0.73 SLC6A2 (0.63) ROCK1SLC6A2MEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0509400-B1 1-(Pyrido[3,4-b]-1,4-oxazinyl-4-yl)-1H-indoles, intermediates and a process for their preparation, and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1996-07-03 EP disclosed
US-5519131-A CYCLIZATION OF HYDROXYALKYLAMINO COMPOUND IN THE PRESENCE OF STRONG BASE SUCH AS SODIUM HYDRIDE OR POTASSIUM TERT-BUTOXIDE HOECHST MARION ROUSSEL INC. (US) 1996-05-21 US disclosed
US-5276156-A Antidepressants, treatment of Alzheimer*s disease HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-01-04 US disclosed
US-5214038-A Cholinesterase inhibitors, antidepressants, cognition activators HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-05-25 US disclosed
EP-0509400-A1 1-(Pyrido[3,4-b]-1,4-oxazinyl-4-yl)-1H-indoles, intermediates and a process for their preparation, and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-10-21 EP disclosed