SCHEMBL8946304

SCHEMBL8946304

O=C(O)c1nc2ccccc2c(F)c1F

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
MAPT P10636 1/20 0.61
DYRK1A Q13627 4/20 0.49
KDM4E B2RXH2 4/20 0.46
PDE10A Q9Y233 2/20 0.46
LMNA P02545 1/20 0.46
DYRK1B Q9Y463 3/20 0.44
CLK1 P49759 2/20 0.44
CDK9 P50750 2/20 0.44
DYRK2 Q92630 2/20 0.44
CLK4 Q9HAZ1 2/20 0.44
CDK5 Q00535 1/20 0.44
CLK2 P49760 1/20 0.44
GSK3B P49841 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
DHODH Q02127 1/20 0.44
ASPH Q12797 1/20 0.43
KDM8 Q8N371 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27775101 0.85 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2MAPTDYRK1AKDM4E
SCHEMBL9258827 0.84 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2MAPTDYRK1AKDM4E
SCHEMBL9258832 0.84 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2MAPTDYRK1AKDM4E
SCHEMBL28156337 0.81 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2MAPTDYRK1AKDM4E
Bicarbonate SCHEMBL10810371 0.78 SMN1; SMN2 (0.42) ALDH1A1SMN1; SMN2MAPTKDM4EPDE10A
SCHEMBL3067398 0.78 ALDH1A1 (0.68) ALDH1A1SMN1; SMN2MAPTDYRK1AKDM4E
SCHEMBL28977964 0.77 SMN1; SMN2 (0.51) ALDH1A1SMN1; SMN2MAPTKDM4ELMNA
SCHEMBL29860539 0.77 ALDH1A1 (1.00) ALDH1A1SMN1; SMN2MAPTDYRK1AKDM4E
SCHEMBL351486 0.77 ALDH1A1 (1.00) ALDH1A1SMN1; SMN2MAPTDYRK1AKDM4E
SCHEMBL8645930 0.77 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2MAPTDYRK1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5493027-A ANTIEPILEPTIC AGENTS, NEUROGENATIVE DISEASES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1996-02-20 US disclosed
WO-1994017042-A1 ANTICONVULSIVE AGENTS AND USES THEREOF BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1994-08-04 WO disclosed
EP-0239992-A1 Process for the preparation of 2,3,4,5-tetrafluorobenzoyl acetates WARNER-LAMBERT COMPANY (US) 1987-10-07 EP disclosed
US-4689423-A Process for the preparation of 2,3,4,5-tetrafluorobenzoyl acetates WARNER-LAMBERT COMPANY (US) 1987-08-25 US disclosed