SCHEMBL8946370

SCHEMBL8946370

CC(C)c1ccc2c(c1)-c1c([nH]c3ccccc13)C2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.53
CA1 P00915 10/20 0.40
CA2 P00918 10/20 0.40
CA4 P22748 10/20 0.40
CA6 P23280 10/20 0.40
DRD2 P14416 4/20 0.38
DRD1 P21728 4/20 0.38
DRD5 P21918 4/20 0.38
DRD3 P35462 4/20 0.38
KDM4E B2RXH2 2/20 0.38
DRD4 P21917 2/20 0.38
MEN1 O00255 1/20 0.38
GMNN O75496 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ADRA1D P25100 1/20 0.38
CYP2C19 P33261 1/20 0.38
ADRA1A P35348 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946421 0.79 CA1 (0.55) CA1CA2CA4CA6DRD2
SCHEMBL8946806 0.79 KIF11 (0.51) KIF11CA1CA2CA4CA6
SCHEMBL8946574 0.79 CA1 (0.65) CA1CA2CA4CA6DRD2
SCHEMBL4374361 0.78 CA1 (0.56) CA1CA2CA4CA6DRD2
SCHEMBL29370154 0.78 CA1 (0.56) CA1CA2CA4CA6DRD2
SCHEMBL9528181 0.74 KMT2A (0.56) KDM4EMEN1CYP1A2KMT2AHPGD
SCHEMBL8946744 0.70 CA1 (0.63) KIF11CA1CA2CA4CA6
SCHEMBL4898197 0.70 LMNA (0.52) KIF11CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL29940783 0.70 CA1 (0.50) CA1CA2CA4CA6DRD2
SCHEMBL13010630 0.70 KIF11 (0.79) KIF11KDM4EMEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516788-A TREATMENT OF ATHEROSCLEROSIS; ANTIISCHEMIC, ANTICARCINOGENIC AGENTS; ANTICOAGULANTS UNIVERSITY OF BATH (GB) 1996-05-14 US disclosed
EP-0409410-B1 Indenoindole compounds UNIV BATH (GB) 1996-03-20 EP disclosed
US-5185360-A Antioxidants, free radical scavengers UNIVERSITY OF BATH (GB) 1993-02-09 US disclosed
EP-0409410-A1 Indenoindole compounds UNIVERSITY OF BATH (GB) 1991-01-23 EP disclosed
WO-1990015799-A1 INDENOINDOLE COMPOUNDS II UNIVERSITY OF BATH (GB) 1990-12-27 WO disclosed
WO-1990015800-A1 INDENOINDOLE COMPOUNDS UNIVERSITY OF BATH (GB) 1990-12-27 WO disclosed
EP-0404536-A1 Indenoindole compounds I UNIVERSITY OF BATH (GB) 1990-12-27 EP disclosed