SCHEMBL8947409

SCHEMBL8947409

CC(C)Cn1c(=O)n(C(=O)N[C@H]2C[C@H]3CC[C@@H](C2)N3C)c2ccccc21

nearest known ligand 0.80

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 4/20 0.80
HTR3A P46098 3/20 0.80
TMEM97 Q5BJF2 1/20 0.80
SIGMAR1 Q99720 1/20 0.80
CNR2 P34972 1/20 0.49
HTR3E A5X5Y0 2/20 0.48
HTR3B O95264 2/20 0.48
HTR3D Q70Z44 2/20 0.48
HTR3C Q8WXA8 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343281 1.00 HTR4 (0.80) HTR4HTR3ATMEM97SIGMAR1CNR2
SCHEMBL1041383 0.89 HTR4 (1.00) HTR4HTR3ATMEM97SIGMAR1HTR3E
SCHEMBL6669870 0.89 HTR4 (1.00) HTR4HTR3ATMEM97SIGMAR1HTR3E
SCHEMBL7343018 0.88 HTR3A (0.85) HTR4HTR3ATMEM97SIGMAR1CNR2
SCHEMBL9398539 0.88 HTR3A (0.85) HTR4HTR3ATMEM97SIGMAR1CNR2
Hydrochloric Acid SCHEMBL8717464 0.88 HTR4 (0.98) HTR4HTR3ATMEM97SIGMAR1HTR3E
Hydrochloric Acid SCHEMBL29386085 0.88 HTR4 (0.98) HTR4HTR3ATMEM97SIGMAR1HTR3E
Hydrochloric Acid SCHEMBL678218 0.87 HTR4 (0.96) HTR4HTR3ATMEM97SIGMAR1HTR3E
Hydrochloric Acid SCHEMBL9572388 0.87 HTR4 (0.96) HTR4HTR3ATMEM97SIGMAR1HTR3E
SCHEMBL7389967 0.84 HTR4 (0.91) HTR4HTR3ATMEM97SIGMAR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5552408-A Benzimidazoline-2-oxo-1-carboxylic acid derivatives useful as 5-ht receptor antagonists BOEHRINGER INGELHEIM ITALIA S.P.A. (IT) 1996-09-03 US disclosed
US-5358954-A Antiserotonine agent, antiemetic, gastrointestinal disorders BOEHRINGER INGELHEIM ITALIA (IT) 1994-10-25 US disclosed
US-5223511-A Benzimidazoline-2-oxo-1-carboxylic acid compounds useful as 5-HT receptor antagonists BOEHRINGER INGELHEIM ITALIA S.P.A. (IT) 1993-06-29 US disclosed