SCHEMBL8947787

SCHEMBL8947787

O=C(c1ccccc1)C1CCN(CCn2c(=O)sc3cc(CCCCN4CCOCC4)ccc32)CC1

nearest known ligand 0.84

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.58
TMEM97 Q5BJF2 1/20 0.51
KDM4E B2RXH2 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
HTR2A P28223 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947902 0.92 KCNH2 (0.53) SIGMAR1TMEM97
SCHEMBL8948078 0.92 HTR2A (0.55) SIGMAR1TMEM97KDM4ECYP1A2CYP3A4
SCHEMBL8947898 0.90 HTR2A (0.55) SIGMAR1KDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL8948101 0.89 TMEM97 (0.49) SIGMAR1TMEM97
SCHEMBL8947963 0.89 SIGMAR1 (0.50) SIGMAR1TMEM97
SCHEMBL8947881 0.88 SIGMAR1 (0.55) SIGMAR1TMEM97
SCHEMBL8947838 0.88 SIGMAR1 (0.56) SIGMAR1TMEM97
SCHEMBL8947866 0.88 SIGMAR1 (0.56) SIGMAR1TMEM97
SCHEMBL8948029 0.87 SIGMAR1 (0.51) SIGMAR1TMEM97
SCHEMBL8947985 0.86 KDM4E (0.58) SIGMAR1KDM4ECYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed