SCHEMBL8948101

SCHEMBL8948101

O=C(c1ccc(C(F)(F)F)cc1)C1CCN(CCn2c(=O)sc3cc(CCCCN4CCOCC4)ccc32)CC1

nearest known ligand 0.84

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.49
HTR1A P08908 1/20 0.48
SIGMAR1 Q99720 2/20 0.48
CNR2 P34972 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948078 0.91 HTR2A (0.55) TMEM97SIGMAR1CNR2
SCHEMBL8947898 0.90 HTR2A (0.55) SIGMAR1CNR2
SCHEMBL8947902 0.90 KCNH2 (0.53) TMEM97SIGMAR1CNR2
SCHEMBL8947787 0.89 SIGMAR1 (0.58) TMEM97SIGMAR1
SCHEMBL8947963 0.87 SIGMAR1 (0.50) TMEM97SIGMAR1CNR2
SCHEMBL8947881 0.86 SIGMAR1 (0.55) TMEM97SIGMAR1CNR2
SCHEMBL8947935 0.85 HTR2A (0.59) TMEM97HTR1ASIGMAR1
SCHEMBL8947762 0.83 HTR1A (0.66) HTR1ASIGMAR1
SCHEMBL8948106 0.82 HTR2A (0.49) HTR1ASIGMAR1CNR2
SCHEMBL8947985 0.81 KDM4E (0.58) HTR1ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed