SCHEMBL8947973

SCHEMBL8947973

COc1ccc2cccc(C(=O)C3CCN(CCn4c(=O)sc5cc(CCCCN6CCOCC6)ccc54)CC3)c2c1

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.46
HTR1A P08908 1/20 0.42
HTR2C P28335 1/20 0.42
CNR2 P34972 1/20 0.42
TMEM97 Q5BJF2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8948029 0.90 SIGMAR1 (0.51) SIGMAR1TMEM97
SCHEMBL8947963 0.86 SIGMAR1 (0.50) SIGMAR1CNR2TMEM97
SCHEMBL8947883 0.85 SIGMAR1 (0.46) SIGMAR1TMEM97
SCHEMBL8947787 0.81 SIGMAR1 (0.58) SIGMAR1TMEM97
SCHEMBL8948069 0.80 SIGMAR1 (0.49) SIGMAR1TMEM97
SCHEMBL8947902 0.78 KCNH2 (0.53) SIGMAR1CNR2TMEM97
SCHEMBL8948078 0.78 HTR2A (0.55) SIGMAR1HTR2CCNR2TMEM97
SCHEMBL8947881 0.76 SIGMAR1 (0.55) SIGMAR1CNR2TMEM97
SCHEMBL8947898 0.76 HTR2A (0.55) SIGMAR1HTR2CCNR2
SCHEMBL8947866 0.76 SIGMAR1 (0.56) SIGMAR1TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed