SCHEMBL8948026

SCHEMBL8948026

CN(C)CCCc1cccc(NC(=O)NCc2c(-c3ccccc3)c3cc(Cl)ccc3c(=O)n2C)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 7/20 0.49
TACR1 P25103 4/20 0.44
LMNA P02545 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TP53 P04637 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPT P10636 2/20 0.41
MAPK8 P45983 2/20 0.41
KCNA5 P22460 1/20 0.41
KCNH2 Q12809 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CNR1 P21554 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947887 0.90 DPP4 (0.52) DPP4TACR1LMNAMAPTMAPK8
Hydrochloric Acid SCHEMBL8948140 0.90 DPP4 (0.51) DPP4TACR1LMNAMAPTMAPK8
SCHEMBL8947927 0.89 DPP4 (0.49) DPP4TACR1LMNAMEN1KMT2A
SCHEMBL8947984 0.87 DPP4 (0.53) DPP4TACR1LMNAMEN1KMT2A
SCHEMBL8947951 0.87 DPP4 (0.61) DPP4TACR1LMNAMEN1KMT2A
SCHEMBL8947829 0.87 DPP4 (0.53) DPP4TACR1LMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL8947929 0.86 DPP4 (0.52) DPP4TACR1LMNAMEN1KMT2A
SCHEMBL8947968 0.86 DPP4 (0.52) DPP4TACR1LMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL8947893 0.86 DPP4 (0.52) DPP4TACR1LMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL8947831 0.86 DPP4 (0.60) DPP4TACR1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527811-A CALCIUM- AND SUBSTANCE P RECEPTOR-ANTAGONIST ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-18 US disclosed
EP-0634402-A1 Isochinolinone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-01-18 EP disclosed