SCHEMBL8948039

SCHEMBL8948039

COc1ccc(N2CCN(CCCCc3ccc4[nH]c(=O)sc4c3)CC2)c2ccccc12

nearest known ligand 0.81

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 13/20 0.81
HTR2C P28335 9/20 0.81
DRD2 P14416 3/20 0.56
HTR2A P28223 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8787054 0.90 HTR1A (1.00) HTR1AHTR2CDRD2HTR2A
SCHEMBL7761398 0.87 HTR1A (1.00) HTR1AHTR2CDRD2HTR2A
SCHEMBL8948107 0.84 HTR1A (0.73) HTR1AHTR2CDRD2HTR2A
SCHEMBL8786294 0.83 HTR1A (1.00) HTR1AHTR2CDRD2HTR2A
SCHEMBL8947946 0.82 HTR1A (0.79) HTR1AHTR2CDRD2HTR2A
SCHEMBL8947912 0.80 HTR1A (0.85) HTR1AHTR2CDRD2HTR2A
SCHEMBL4891426 0.77 HTR1A (0.75) HTR1AHTR2CDRD2HTR2A
SCHEMBL4888935 0.77 HTR1A (0.63) HTR1AHTR2CDRD2HTR2A
SCHEMBL8948002 0.77 HTR1A (0.87) HTR1AHTR2CDRD2HTR2A
Hydrochloric Acid SCHEMBL7099408 0.76 HTR1A (0.62) HTR1AHTR2CDRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed