SCHEMBL8948002

SCHEMBL8948002

O=c1[nH]c2ccc(CCCN3CCN(c4ccccc4)CC3)cc2s1

nearest known ligand 0.87

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 9/20 0.87
HTR2C P28335 8/20 0.87
DRD2 P14416 4/20 0.64
SIGMAR1 Q99720 4/20 0.58
HTR2A P28223 1/20 0.57
HTR7 P34969 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947912 0.97 HTR1A (0.85) HTR1AHTR2CDRD2SIGMAR1HTR2A
SCHEMBL8948209 0.93 HTR1A (1.00) HTR1AHTR2CDRD2HTR2A
SCHEMBL8785423 0.86 HTR1A (0.69) HTR1AHTR2CDRD2SIGMAR1HTR2A
SCHEMBL7756727 0.84 HTR1A (0.64) HTR1AHTR2CDRD2HTR2A
SCHEMBL467277 0.83 HTR1A (0.61) HTR1AHTR2CDRD2SIGMAR1HTR2A
SCHEMBL7756745 0.83 HTR1A (0.63) HTR1AHTR2CDRD2HTR2A
SCHEMBL8786197 0.83 HTR1A (0.81) HTR1AHTR2CDRD2SIGMAR1HTR2A
SCHEMBL7761398 0.83 HTR1A (1.00) HTR1AHTR2CDRD2HTR2AHTR7
SCHEMBL8947948 0.83 HTR1A (1.00) HTR1AHTR2CDRD2SIGMAR1HTR2A
SCHEMBL7763020 0.82 HTR1A (0.62) HTR1AHTR2CDRD2SIGMAR1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed