SCHEMBL8948142

SCHEMBL8948142

CN(C)Cc1ccc(NC(=O)NCc2c(-c3ccccc3)c3cc(Cl)ccc3c(=O)n2C)cc1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LSS P48449 1/20 0.53
DPP4 P27487 7/20 0.53
TACR1 P25103 4/20 0.49
KCNA5 P22460 1/20 0.48
KCNH2 Q12809 1/20 0.48
MAPK8 P45983 6/20 0.46
SLC2A1 P11166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947887 0.91 DPP4 (0.52) LSSDPP4TACR1KCNA5KCNH2
Hydrochloric Acid SCHEMBL8948140 0.91 DPP4 (0.51) LSSDPP4TACR1KCNA5KCNH2
SCHEMBL8947848 0.87 DPP4 (0.57) DPP4TACR1MAPK8
SCHEMBL8947888 0.87 DPP4 (0.54) DPP4TACR1KCNA5KCNH2MAPK8
SCHEMBL8947988 0.86 DPP4 (0.56) DPP4TACR1MAPK8
SCHEMBL8947983 0.86 DPP4 (0.56) DPP4TACR1MAPK8
SCHEMBL8947680 0.86 DPP4 (0.53) DPP4TACR1KCNA5KCNH2MAPK8
SCHEMBL8947987 0.85 DPP4 (0.54) DPP4TACR1MAPK8
SCHEMBL8947829 0.84 DPP4 (0.53) DPP4TACR1KCNA5KCNH2MAPK8
Hydrochloric Acid SCHEMBL8947893 0.83 DPP4 (0.52) DPP4TACR1KCNA5KCNH2MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527811-A CALCIUM- AND SUBSTANCE P RECEPTOR-ANTAGONIST ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-18 US disclosed
EP-0634402-A1 Isochinolinone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-01-18 EP disclosed