SCHEMBL8947888

SCHEMBL8947888

CN(C)Cc1cccc(CNC(=O)NCc2c(-c3ccccc3)c3cc(Cl)ccc3c(=O)n2C)c1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 9/20 0.54
KCNA5 P22460 1/20 0.49
KCNH2 Q12809 1/20 0.49
TACR1 P25103 8/20 0.48
ACP1 P24666 1/20 0.41
MAPK8 P45983 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947887 0.91 DPP4 (0.52) DPP4KCNA5KCNH2TACR1ACP1
Hydrochloric Acid SCHEMBL8948140 0.90 DPP4 (0.51) DPP4KCNA5KCNH2TACR1ACP1
SCHEMBL8948142 0.87 LSS (0.53) DPP4KCNA5KCNH2TACR1MAPK8
SCHEMBL8947680 0.83 DPP4 (0.53) DPP4KCNA5KCNH2TACR1MAPK8
SCHEMBL8948186 0.82 DPP4 (0.50) DPP4KCNA5KCNH2TACR1MAPK8
Hydrochloric Acid SCHEMBL8948118 0.82 TACR1 (0.50) KCNA5KCNH2TACR1
SCHEMBL8947984 0.81 DPP4 (0.53) DPP4TACR1MAPK8
SCHEMBL8948026 0.81 DPP4 (0.49) DPP4KCNA5KCNH2TACR1MAPK8
Hydrochloric Acid SCHEMBL8947929 0.81 DPP4 (0.52) DPP4TACR1MAPK8
SCHEMBL8948130 0.80 DPP4 (0.52) DPP4TACR1MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527811-A CALCIUM- AND SUBSTANCE P RECEPTOR-ANTAGONIST ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-18 US disclosed
EP-0634402-A1 Isochinolinone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-01-18 EP disclosed