SCHEMBL8948258

SCHEMBL8948258

O=C1OC(CO)CN1Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 12/20 0.54
SIRT1 Q96EB6 1/20 0.46
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
CALML3 P27482 1/20 0.44
FADS1 O60427 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12356902 1.00 GRM2 (0.54) GRM2SIRT1MAOAMAOBHPGD
SCHEMBL2832723 0.86 GRM2 (0.55) GRM2SIRT1HPGDTSHR
SCHEMBL11744593 0.86 GRM2 (0.63) GRM2SIRT1HPGDTSHR
SCHEMBL2836661 0.86 GRM2 (0.55) GRM2SIRT1HPGDTSHR
SCHEMBL15757602 0.85 MAPK1 (0.46) GRM2MAOAMAOBHPGDCALML3
SCHEMBL20485430 0.85 GRM2 (0.45) GRM2MAOAMAOB
SCHEMBL15758259 0.85 MAOA (0.49) GRM2MAOAMAOB
SCHEMBL15757524 0.85 GRM2 (0.60) GRM2CALML3FADS1
SCHEMBL14662038 0.85 MAPK1 (0.46) GRM2MAOAMAOBHPGDCALML3
SCHEMBL1972447 0.85 MAPK1 (0.46) GRM2MAOAMAOBHPGDCALML3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-8183782-A None JP disclosed
CN-112409286-B Synthesis method of N-substituted phenyl-5-hydroxymethyl-2-oxazolidinone 杭州迪克科技有限公司 2022-08-05 CN disclosed
CN-112409286-A Synthesis method of N-substituted phenyl-5-hydroxymethyl-2-oxazolidinone 杭州迪克科技有限公司 2021-02-26 CN disclosed
US-9464062-B2 Disubstituted oxazolidin-2-ones 5-hydroxytryptamine receptor 2B activity modulators Temple University—Of the Commonwealth System of Higher Education (US) 2016-10-11 US disclosed
US-9464062-B2 Disubstituted oxazolidin-2-ones 5-hydroxytryptamine receptor 2B activity modulators Temple University—Of the Commonwealth System of Higher Education (US) 2016-10-11 US disclosed
US-9464062-B2 Disubstituted oxazolidin-2-ones 5-hydroxytryptamine receptor 2B activity modulators Temple University—Of the Commonwealth System of Higher Education (US) 2016-10-11 US disclosed
US-20150291539-A1 DISUBSTITUTED OXAZOLIDIN-2-ONES 5-HYDROXYTRYPTAMINE RECEPTOR 2B ACTIVITY MODULATORS TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2015-10-15 US disclosed
US-20150291539-A1 DISUBSTITUTED OXAZOLIDIN-2-ONES 5-HYDROXYTRYPTAMINE RECEPTOR 2B ACTIVITY MODULATORS TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2015-10-15 US disclosed
US-20150291539-A1 DISUBSTITUTED OXAZOLIDIN-2-ONES 5-HYDROXYTRYPTAMINE RECEPTOR 2B ACTIVITY MODULATORS TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2015-10-15 US disclosed
WO-2014085413-A1 DISUBSTITUTED OXAZOLIDIN-2-ONES 5-HYDROXYTRYPTAMINE RECEPTOR 2B ACTIVITY MODULATORS TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2014-06-05 WO disclosed
JP-H08183782-A METHOD FOR CRYSTALLIZING 4-BENZYL-5-HYDROXYMETHYLOXAZOLIDIN-2-ONE KANEGAFUCHI CHEM IND CO LTD 1996-07-16 JP disclosed
US-4886794-A ANTIHISTAMINES, ANTIALLERGENS A. H. ROBINS COMPANY, INCORPORATED (US) 1989-12-12 US disclosed
EP-0291244-A1 Cyclic carbamate derivatives A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1988-11-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150291539-A1 DISUBSTITUTED OXAZOLIDIN-2-ONES 5-HYDROXYTRYPTAMINE RECEPTOR 2B ACTIVITY MODULATORS HTR2B, TPH2, HTR2C GRM2 77/4885SIRT1 2310/4885MAOA 86/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.