SCHEMBL8949093

SCHEMBL8949093

CCOC(=O)c1cc(-c2ccc(C#N)cc2)nnc1Cl

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 10/20 0.70
KDM4E B2RXH2 3/20 0.52
ALDH1A1 P00352 3/20 0.52
HPGD P15428 3/20 0.52
GAA P10253 1/20 0.52
SMN1; SMN2 Q16637 3/20 0.45
NPSR1 Q6W5P4 2/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
MEN1 O00255 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 1/20 0.45
ELANE P08246 1/20 0.43
ALPL P05186 1/20 0.43
HSD17B10 Q99714 1/20 0.42
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5899777 0.82 CASP1 (1.00) CASP1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL8949196 0.80 CASP1 (0.77) CASP1ALDH1A1HPGDCYP2C9HSD17B10
SCHEMBL7275356 0.77 KDM4E (0.51) KDM4EALDH1A1HPGDGAASMN1; SMN2
SCHEMBL7276252 0.76 HPGD (0.57) KDM4EALDH1A1HPGDGAASMN1; SMN2
SCHEMBL30051126 0.74 CASP1 (0.62) CASP1KDM4EALDH1A1TSHRMAPK1
SCHEMBL140932 0.74 CASP1 (0.62) CASP1KDM4EALDH1A1TSHRMAPK1
SCHEMBL7992182 0.73 CYP4F2 (0.48) KDM4EALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL27944765 0.73 CYP4F2 (0.58) KDM4EALDH1A1HPGDGAASMN1; SMN2
SCHEMBL2650679 0.73 KDM4E (0.48) KDM4EALDH1A1HPGDGAASMN1; SMN2
SCHEMBL8949195 0.73 SMN1; SMN2 (0.59) KDM4EALDH1A1HPGDGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed