SCHEMBL8949196

SCHEMBL8949196

N#Cc1ccc(-c2cc(C(=O)O)c(Cl)nn2)cc1

nearest known ligand 0.77

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 14/20 0.77
MAOB P27338 1/20 0.45
EIF4E P06730 1/20 0.45
GABRA1 P14867 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
RPA1 P27694 1/20 0.41
XDH P47989 1/20 0.40
SLC22A12 Q96S37 1/20 0.40
PTGES O14684 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ALOX5 P09917 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CASP7 P55210 1/20 0.40
HIF1A Q16665 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL580314 0.81 CASP1 (0.76) CASP1ALDH1A1HIF1AHSD17B10
SCHEMBL8949093 0.80 CASP1 (0.70) CASP1ALDH1A1CYP2C9HPGDHSD17B10
SCHEMBL27225888 0.80 CASP1 (0.56) CASP1ALDH1A1HSD17B10
SCHEMBL30850823 0.80 CASP1 (0.56) CASP1ALDH1A1HSD17B10
SCHEMBL30448360 0.73 DHODH (0.61) CASP1EIF4E
SCHEMBL7277324 0.72 CASP1 (0.46) CASP1RPA1XDHSLC22A12
SCHEMBL22506701 0.72 KDM4E (0.47) CASP1EIF4EGABRA1GABRG2GABRB3
SCHEMBL6727952 0.72 CASP1 (0.56) CASP1MAOBGABRA1GABRG2GABRB3
SCHEMBL1897930 0.71 DHODH (0.74) ALDH1A1HPGD
SCHEMBL15904177 0.70 DHODH (0.76) ALDH1A1HPGDHIF1AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed