SCHEMBL8949128

SCHEMBL8949128

CN(CC(=O)O)C(=O)CNC(=O)c1cc(-c2ccc(C(=N)N)cc2)nn(C)c1=O

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 3/20 0.35
ITGB3 P05106 9/20 0.35
ITGA2B P08514 9/20 0.35
RXFP1 Q9HBX9 1/20 0.35
HPGD P15428 1/20 0.34
F2 P00734 2/20 0.33
KLKB1 P03952 1/20 0.33
PRSS1 P07477 1/20 0.33
TMPRSS15 P98073 1/20 0.33
CGAS Q8N884 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8949032 0.91 RXFP1 (0.37) PHGDHITGB3ITGA2BRXFP1HPGD
SCHEMBL8949398 0.85 ITGB3 (0.40) PHGDHITGB3ITGA2BF2KLKB1
SCHEMBL8949239 0.82 ITGB3 (0.45) ITGB3ITGA2B
SCHEMBL8949379 0.82 HPGD (0.38) PHGDHITGB3ITGA2BHPGDKLKB1
SCHEMBL8949063 0.81 ITGB3 (0.47) ITGB3ITGA2B
SCHEMBL8949221 0.80 HPGD (0.37) PHGDHITGB3ITGA2BHPGD
SCHEMBL8949033 0.80 ITGB3 (0.51) ITGB3ITGA2B
SCHEMBL8949233 0.79 HPGD (0.40) PHGDHITGB3ITGA2BHPGDF2
SCHEMBL8949188 0.79 ALDH1A1 (0.38) PHGDHITGB3ITGA2BHPGDF2
Hydrochloric Acid SCHEMBL8949365 0.79 F2 (0.39) ITGB3ITGA2BRXFP1HPGDF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed