SCHEMBL8949131

SCHEMBL8949131

COC(=O)[C@H]1CC[C@@H](NC(=O)c2cc(-c3ccc(C(=N)N)cc3)nn(C)c2=O)CC1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.42
CNR2 P34972 5/20 0.42
CNR1 P21554 4/20 0.42
F2 P00734 11/20 0.41
ST14 Q9Y5Y6 8/20 0.41
PRSS1 P07477 5/20 0.41
PRSS2 P07478 5/20 0.41
PRSS3 P35030 5/20 0.41
PLG P00747 2/20 0.41
F10 P00742 3/20 0.40
KLK7 P49862 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TMPRSS15 P98073 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8949034 1.00 CFTR (0.42) CFTRCNR2CNR1F2ST14
SCHEMBL8949277 0.91 CNR2 (0.46) CNR2CNR1F2ST14PRSS1
SCHEMBL8949148 0.91 CNR2 (0.46) CNR2CNR1F2ST14PRSS1
SCHEMBL8949056 0.89 CNR2 (0.41) CFTRCNR2CNR1KLK7HPGD
SCHEMBL8949258 0.89 CNR2 (0.41) CFTRCNR2CNR1KLK7HPGD
Hydrochloric Acid SCHEMBL8949181 0.88 CNR2 (0.46) CFTRCNR2CNR1F2ST14
Hydrochloric Acid SCHEMBL8949338 0.87 CNR2 (0.45) CFTRCNR2CNR1F2ST14
Hydrochloric Acid SCHEMBL8949314 0.87 F2 (0.36) CFTRCNR2F2ST14PRSS1
Hydrochloric Acid SCHEMBL8949274 0.86 CNR1 (0.44) CFTRCNR2CNR1F2ST14
Hydrochloric Acid SCHEMBL8949113 0.86 TMPRSS15 (0.41) CFTRCNR2CNR1F2ST14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed