SCHEMBL8949200

SCHEMBL8949200

N#Cc1ccc(-c2cc(C(=O)O)c(=O)n(CC(=O)N3CCOCC3)n2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.46
KDM4E B2RXH2 4/20 0.45
HSD17B10 Q99714 2/20 0.45
POLB P06746 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
MKNK1 Q9BUB5 2/20 0.43
MKNK2 Q9HBH9 2/20 0.43
PRKDC P78527 1/20 0.42
ALDH1A1 P00352 5/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
SCN7A Q01118 2/20 0.41
KCNH2 Q12809 2/20 0.41
USP2 O75604 1/20 0.41
TP53 P04637 1/20 0.41
ALOX15 P16050 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
NPC1 O15118 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8949298 0.87 KDM4E (0.47) TSHRKDM4EHSD17B10POLBCYP3A4
SCHEMBL9260471 0.80 CNR2 (0.41) POLBHPGDEGLN1
SCHEMBL28300713 0.76 MEN1 (0.51) KDM4EHSD17B10POLBALDH1A1SMN1; SMN2
SCHEMBL8949294 0.76 CNR1 (0.46) POLBSMN1; SMN2GAAMEN1KMT2A
SCHEMBL29784613 0.75 TSHR (0.59) TSHRKDM4EHSD17B10POLBCYP3A4
SCHEMBL23909112 0.73 S1PR2 (0.45) ALDH1A1SCN7AKCNH2TP53GAA
SCHEMBL7275259 0.72 PHGDH (0.48) KDM4EALDH1A1GAAHPGDMEN1
SCHEMBL8949199 0.69 ITGB3 (0.43) TSHRKDM4EHSD17B10POLBCYP3A4
SCHEMBL9571672 0.68 ITGB3 (0.38) TSHRKDM4EHSD17B10POLBCYP3A4
SCHEMBL23915287 0.67 S1PR2 (0.45) KDM4EPOLBALDH1A1SCN7AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed