SCHEMBL8949305

SCHEMBL8949305

FC(F)(F)c1ccc(CNCCCn2ccnc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.59
HMOX1 P09601 1/20 0.53
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
NPC1 O15118 1/20 0.49
QPCT Q16769 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CYP19A1 P11511 1/20 0.48
LMNA P02545 1/20 0.46
ATP4A P20648 1/20 0.46
ATP4B P51164 1/20 0.46
VEGFA P15692 1/20 0.46
EGLN1 Q9GZT9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8949252 0.99 NOS1 (0.57) NOS1HMOX1CYP1A2CYP3A4CYP2D6
SCHEMBL3181153 0.89 SMN1; SMN2 (0.57) HMOX1SMN1; SMN2NPC1QPCTCYP19A1
SCHEMBL14416010 0.86 SMN1; SMN2 (0.56) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL14416009 0.85 CYP19A1 (0.67) SMN1; SMN2QPCTCYP19A1LMNA
Hydrochloric Acid SCHEMBL8949368 0.83 NOS1 (0.48) NOS1HMOX1SMN1; SMN2QPCTL3MBTL1
SCHEMBL8443968 0.82 HMOX1 (0.65) NOS1HMOX1SMN1; SMN2QPCTCYP19A1
SCHEMBL6571544 0.82 CYP1A2 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL2475754 0.82 QPCT (0.67) CYP1A2CYP3A4CYP2D6SMN1; SMN2QPCT
SCHEMBL3166171 0.81 SMN1; SMN2 (0.53) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL10283707 0.81 NOS1 (0.67) NOS1HMOX1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1037511-C Therapeutic agents BOOTS CO PLC (GB) 1998-02-25 CN disclosed
US-5547972-A 1-(ARLALKYLAMINOALKYL) IMIDAZOLE DERIVATIVES THE BOOTS COMPANY PLC (GB) 1996-08-20 US disclosed
EP-0618907-A1 1-(ARYLALKYL-AMINOALKYL)IMIDAZOLE DERIVATIVES, PROCESSES OF PREPARATION AND USE AS THERAPEUTICAL AGENTS Knoll AG (DE) 1994-10-12 EP disclosed
WO-1993013075-A1 1-(ARYLALKYL-AMINOALKYL)IMIDAZOLE DERIVATIVES, PROCESSES OF PREPARATION AND USE AS THERAPEUTICAL AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed