SCHEMBL8949321

SCHEMBL8949321

COC(=O)CC1CCN(C(=O)c2ncc(-c3ccc(C(=N)NC(=O)OC)cc3)cn2)CC1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.37
ITGB3 P05106 8/20 0.36
ITGA2B P08514 8/20 0.36
HTR2B P41595 2/20 0.36
GPR119 Q8TDV5 2/20 0.35
POLB P06746 1/20 0.34
MELK Q14680 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ABL1 P00519 1/20 0.34
BCR P11274 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8407957 0.89 POLB (0.43) HRH3ITGB3ITGA2BHTR2BPOLB
Hydrochloric Acid SCHEMBL8949325 0.87 ITGB3 (0.45) ITGB3ITGA2B
SCHEMBL8410914 0.82 ITGB3 (0.42) HRH3ITGB3ITGA2BPOLBALDH1A1
SCHEMBL8949271 0.82 HTR2B (0.41) ITGB3ITGA2BHTR2BMELK
SCHEMBL8407952 0.80 ITGB3 (0.49) ITGB3ITGA2BPOLBALDH1A1SMN1; SMN2
SCHEMBL9568137 0.79 HRH3 (0.39) HRH3ITGB3ITGA2BHTR2BPOLB
SCHEMBL9568130 0.79 POLB (0.41) HRH3ITGB3ITGA2BHTR2BPOLB
SCHEMBL8409563 0.79 SMN1; SMN2 (0.49) HRH3HTR2BPOLBALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL8949278 0.79 ITGB3 (0.41) ITGB3ITGA2B
SCHEMBL9568214 0.79 HRH3 (0.39) HRH3ITGB3ITGA2BHTR2BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed