SCHEMBL8949698

SCHEMBL8949698

Cc1nc(C)c(CO)c(-c2ccc(F)cc2)c1CO

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GCGR P47871 15/20 0.56
PRKAA2 P54646 1/20 0.44
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
DPP4 P27487 1/20 0.39
USP7 Q93009 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6955413 0.87 GCGR (0.49) GCGRPRKAA2MEN1KMT2A
SCHEMBL8949777 0.86 GCGR (0.74) GCGR
SCHEMBL9263291 0.81 GCGR (0.65) GCGRNPC1RAB9A
SCHEMBL6957028 0.79 GCGR (0.50) GCGRNPC1RAB9A
SCHEMBL7557523 0.79 GCGR (0.47) GCGRDPP4
SCHEMBL2648588 0.78 GCGR (0.86) GCGR
SCHEMBL6956576 0.77 GCGR (0.46) GCGRMEN1NPC1RAB9AKMT2A
SCHEMBL8949822 0.77 GCGR (0.88) GCGR
SCHEMBL10656158 0.77 KDM4E (0.59) GCGRPRKAA2
SCHEMBL2648917 0.75 GCGR (0.86) GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5502057-A Polysubstituted pyridines useful for treating lipoproteinanaemia and arteriosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1996-03-26 US disclosed
US-5470982-A Disubstituted pyridines BAYER AKTIENGESELLSCHAFT (DE) 1995-11-28 US disclosed
EP-0325129-B1 Disubstituted pyridines BAYER AG (DE) 1994-09-07 EP disclosed
US-5173495-A 7-[(2,6-dialkyl-4-furyl or thienyl-pyridyl)]-3,5-di-(dihydroxy-6-enoates) useful for treating circulatory diseases BAYER AKTIENGESELLSCHAFT (DE) 1992-12-22 US disclosed
US-4968689-A Certain 2,6-diisopropyl-4-(4-fluoro-phenyl)-3,5-bis-dimethyl-3',5'-dihydroxy-hept-6-enoate-pyridine derivatives useful for treating lipoproteinaemia and arteriosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1990-11-06 US disclosed
CN-1034716-A Disubstituted pyridines and preparation method thereof BAYER AG (DE) 1989-08-16 CN disclosed
EP-0325129-A2 Disubstituted pyridines BAYER AG (DE) 1989-07-26 EP disclosed