SCHEMBL8950255

SCHEMBL8950255

NS(=O)(=O)c1cc2c(s1)S(=O)(=O)CCN2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CA2 P00918 20/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428610 0.81 CA2 (0.68) CA2
SCHEMBL9429746 0.76 CA2 (0.62) CA2
Hydrochloric Acid SCHEMBL9429811 0.75 CA2 (0.61) CA2
SCHEMBL9682149 0.74 CA2 (1.00) CA2
SCHEMBL9682704 0.73 CA2 (0.72) CA2
Hydrochloric Acid SCHEMBL9429322 0.72 CA2 (0.60) CA2
Hydrochloric Acid SCHEMBL9429319 0.72 CA2 (0.60) CA2
Hydrochloric Acid SCHEMBL9429791 0.72 CA2 (0.60) CA2
SCHEMBL10513455 0.70 CA2 (1.00) CA2
SCHEMBL10514227 0.69 CA2 (1.00) CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0479480-A2 Substituted thieno(2,3-B)(1,4)thiazine-6-sulfonamides as antiglaucoma agents MERCK & CO. INC. (US) 1992-04-08 EP claimed
US-5093332-A SUBSTITUTED THIENO(2,3-B)(1,4)THIAZINE-6-SULFONAMIDES AS ANTIGLAUCOMA AGENTS MERCK & CO., INC. (US) 1992-03-03 US claimed
US-5538966-A ENZYME INHIBITORS FOR TREATMENT OF GLAUCOMA ALCON LABORATORIES, INC. (US) 1996-07-23 US disclosed
WO-1995019981-A1 THIENOTHIAZINE SULFONAMIDE DERIVATIVES PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS CARBONIC ANHYDRASE INHIBITORS ALCON LABORATORIES, INC. (US) 1995-07-27 WO disclosed
EP-0479480-A2 Substituted thieno(2,3-B)(1,4)thiazine-6-sulfonamides as antiglaucoma agents MERCK & CO. INC. (US) 1992-04-08 EP disclosed
US-5093332-A SUBSTITUTED THIENO(2,3-B)(1,4)THIAZINE-6-SULFONAMIDES AS ANTIGLAUCOMA AGENTS MERCK & CO., INC. (US) 1992-03-03 US disclosed