SCHEMBL8952917

SCHEMBL8952917

COP(=O)(C=Cc1c(C2CC2)nc(-c2ccccc2)c(C)c1-c1ccc(F)cc1)C[C@H](CC(=O)O)O[Si](c1ccccc1)(c1ccccc1)C(C)(C)C

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.41
NR4A2 P43354 1/20 0.41
PDE4D Q08499 1/20 0.41
RXRA P19793 2/20 0.38
HMGCR P04035 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8953328 0.89 CTSA (0.32)
SCHEMBL8952769 0.89 ESR1 (0.39) HMGCR
SCHEMBL8952778 0.89 ESR1 (0.39) HMGCR
SCHEMBL8953306 0.89 CTSA (0.32)
SCHEMBL8952873 0.85 NR1I2 (0.51) NR1I2NR4A2PDE4DRXRAHMGCR
SCHEMBL8952914 0.84 NR1I2 (0.33) NR1I2NR4A2PDE4D
SCHEMBL8952807 0.83
SCHEMBL8953217 0.81 ESR1 (0.41) HMGCR
SCHEMBL8953196 0.81 ESR1 (0.41) HMGCR
SCHEMBL9562809 0.80 HMGCR (0.45) NR1I2PDE4DHMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed
EP-0444533-A2 Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1991-09-04 EP disclosed