SCHEMBL8952914

SCHEMBL8952914

C=C(c1c(C2CC2)nc(-c2ccccc2)c(C)c1-c1ccc(F)cc1)P(=O)(C[C@H](CC(=O)O)O[Si](c1ccccc1)(c1ccccc1)C(C)(C)C)OC

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.33
NR4A2 P43354 1/20 0.33
PDE4D Q08499 1/20 0.33
PRKAA2 P54646 1/20 0.32
CTSA P10619 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8952869 0.85 NR1I2 (0.42) NR1I2NR4A2PDE4D
SCHEMBL8952917 0.84 NR1I2 (0.41) NR1I2NR4A2PDE4D
SCHEMBL8952807 0.83
SCHEMBL8952921 0.82 NR1I2 (0.33) NR1I2NR4A2PDE4DPRKAA2
SCHEMBL8952925 0.82 NR1I2 (0.33) NR1I2NR4A2PDE4DPRKAA2
SCHEMBL9562803 0.80 HMGCR (0.34) CTSA
SCHEMBL9562819 0.80 HMGCR (0.34) CTSA
SCHEMBL8952769 0.75 ESR1 (0.39)
SCHEMBL8953306 0.75 CTSA (0.32) CTSA
SCHEMBL8952778 0.75 ESR1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed