SCHEMBL8954166

SCHEMBL8954166

CC(C)C1CCN(C(N)=O)C1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 8/20 0.39
DPP7 Q9UHL4 3/20 0.39
DPP8 Q6V1X1 2/20 0.39
DPP9 Q86TI2 2/20 0.39
CPN1 P15169 1/20 0.38
CPB2 Q96IY4 1/20 0.38
GAA P10253 1/20 0.37
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
ALOX5 P09917 1/20 0.34
PDE4B Q07343 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1109055 0.88 CPN1 (0.40) DPP4DPP7DPP8DPP9CPN1
SCHEMBL20756331 0.83 CHRNB2 (0.38) CPN1CPB2ALOX5
SCHEMBL15837592 0.82 PIK3CD (0.38) DPP4DPP7DPP8DPP9CPN1
SCHEMBL15837591 0.82 PIK3CD (0.38) DPP4DPP7DPP8DPP9CPN1
SCHEMBL679537 0.82 PIK3CD (0.38) DPP4DPP7DPP8DPP9CPN1
SCHEMBL13035374 0.82 CPN1 (0.38) DPP4DPP7DPP8DPP9CPN1
SCHEMBL25961563 0.80 DPP4 (0.41) DPP4DPP7DPP8DPP9CPN1
SCHEMBL16999004 0.80 CHRNB2 (0.46) DPP4DPP7DPP8DPP9MEN1
SCHEMBL10232854 0.80 CPN1 (0.37) DPP4DPP7DPP8DPP9CPN1
SCHEMBL18074021 0.80 CHRNB2 (0.46) DPP4DPP7DPP8DPP9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240182467-A1 INHIBITORS OF RAF KINASES Pierre Fabre Médicament (FR) 2024-06-06 US disclosed
US-11814384-B2 Inhibtors of Raf kinases KINNATE BIOPHARMA INC. (US) 2023-11-14 US disclosed
US-11661410-B2 Tricyclic compounds as histone methyltransferase inhibitors GLOBAL BLOOD THERAPEUTICS, INC. (US) 2023-05-30 US disclosed
US-11661410-B2 Tricyclic compounds as histone methyltransferase inhibitors GLOBAL BLOOD THERAPEUTICS, INC. (US) 2023-05-30 US disclosed
US-20230002351-A1 TRICYCLIC COMPOUNDS AS HISTONE METHYLTRANSFERASE INHIBITORS GLOBAL BLOOD THERAPEUTICS, INC. 2023-01-05 US disclosed
CN-109096274-B Biaryl compounds useful in the treatment of human oncological, neurological and immunological diseases 比奥根MA公司 2022-07-01 CN disclosed
CN-109096274-A It can be used for treating the aryl-linking compound of human tumor, neurology and amynologic disease 比奥根MA公司 2018-12-28 CN disclosed
CN-108947913-A It can be used for treating the aryl-linking compound of human tumor, neurology and amynologic disease 比奥根MA公司 2018-12-07 CN disclosed
CN-106459002-B Biaryl compounds useful in the treatment of human oncological, neurological and immunological diseases 比奥根MA公司 2018-08-21 CN disclosed
US-20180093973-A1 BIARYL INHIBITORS OF BRUTON'S TYROSINE KINASE BIOGEN MA INC. 2018-04-05 US disclosed
CN-106459002-A Biaryl compounds useful in the treatment of human oncological, neurological and immunological diseases 比奥根MA公司 2017-02-22 CN disclosed
US-8188085-B2 Antifungal agents MERCK SHARP & DOHME CORP. (US) 2012-05-29 US disclosed
US-20100113439-A1 Antifungal agents MERCK & CO., INC. (US) 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240182467-A1 INHIBITORS OF RAF KINASES BRAF, RAF1, ARAF DPP4 3912/4885DPP7 2870/4885DPP8 2863/4885
US-20180093973-A1 BIARYL INHIBITORS OF BRUTON'S TYROSINE KINASE ABL1, BTK, LYN DPP4 3722/4885DPP7 2591/4885DPP8 3155/4885
US-20230002351-A1 TRICYCLIC COMPOUNDS AS HISTONE METHYLTRANSFERASE INHIBITORS EHMT1, EHMT2, BMI1 DPP4 1075/4885DPP7 846/4885DPP8 610/4885
US-11661410-B2 Tricyclic compounds as histone methyltransferase inhibitors EHMT1, EHMT2, BMI1 DPP4 1075/4885DPP7 846/4885DPP8 610/4885
US-20100113439-A1 Antifungal agents GMDS, GBA3, UGGT1 DPP4 221/4885DPP7 187/4885DPP8 179/4885
US-11814384-B2 Inhibtors of Raf kinases RAF1, BRAF, ARAF DPP4 4369/4885DPP7 3284/4885DPP8 2799/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.