SCHEMBL8955489

SCHEMBL8955489

CCOC(=O)C1=C(C(C)C)NC(C(C)C)=C(C(=O)OCC)C1c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.63
KDM4E B2RXH2 6/20 0.59
GAA P10253 2/20 0.59
CACNA1D Q01668 3/20 0.54
CACNA1F O60840 1/20 0.54
CACNA1S Q13698 1/20 0.54
CACNA1C Q13936 1/20 0.54
ALDH1A1 P00352 6/20 0.52
TSHR P16473 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
ABCC1 P33527 1/20 0.51
HPGD P15428 3/20 0.50
DHFR P00374 1/20 0.50
SIRT3 Q9NTG7 1/20 0.50
LMNA P02545 1/20 0.50
HSD17B10 Q99714 1/20 0.50
MEN1 O00255 2/20 0.48
MAPT P10636 2/20 0.48
KMT2A Q03164 2/20 0.48
XBP1 P17861 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2647704 0.86 CACNA1F (0.56) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL27310185 0.84 CACNA1F (0.52) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL2648365 0.83 PTPN1 (0.60) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL9270856 0.82 CACNA1D (0.45) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL8949608 0.82 EPHX2 (0.51) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL3027412 0.82 ADORA3 (0.89) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL11669396 0.81 ADORA3 (0.68) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL9359378 0.81 ADORA3 (0.47) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL8950009 0.81 CACNA1F (0.46) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL2662903 0.80 CACNA1F (0.50) ADORA3KDM4EGAACACNA1DCACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5502057-A Polysubstituted pyridines useful for treating lipoproteinanaemia and arteriosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1996-03-26 US disclosed
US-5470982-A Disubstituted pyridines BAYER AKTIENGESELLSCHAFT (DE) 1995-11-28 US disclosed
US-5173495-A 7-[(2,6-dialkyl-4-furyl or thienyl-pyridyl)]-3,5-di-(dihydroxy-6-enoates) useful for treating circulatory diseases BAYER AKTIENGESELLSCHAFT (DE) 1992-12-22 US disclosed
US-4968689-A Certain 2,6-diisopropyl-4-(4-fluoro-phenyl)-3,5-bis-dimethyl-3',5'-dihydroxy-hept-6-enoate-pyridine derivatives useful for treating lipoproteinaemia and arteriosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1990-11-06 US disclosed