SCHEMBL8959513

SCHEMBL8959513

CCc1cn(CC(C)O)c2cc(Cl)c(F)cc12

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ICMT O60725 7/20 0.45
HTR2A P28223 3/20 0.39
HTR2C P28335 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
HTR2B P41595 1/20 0.39
KCNH2 Q12809 1/20 0.36
PIM1 P11309 4/20 0.34
PIM2 Q9P1W9 3/20 0.34
GSK3A P49840 1/20 0.34
PIM3 Q86V86 1/20 0.34
GPR84 Q9NQS5 1/20 0.33
SLC5A2 P31639 1/20 0.32
SLC1A3 P43003 1/20 0.32
SLC1A2 P43004 1/20 0.32
SLC1A1 P43005 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8959510 1.00 ICMT (0.45) ICMTHTR2AHTR2CCYP1A2CYP3A4
SCHEMBL9234274 0.86 HTR2C (0.54) ICMTHTR2AHTR2CCYP1A2CYP3A4
SCHEMBL8959735 0.83 HTR2A (0.41) ICMTHTR2AHTR2CCYP1A2CYP3A4
SCHEMBL8959726 0.83 HTR2A (0.41) ICMTHTR2AHTR2CCYP1A2CYP3A4
Fumaric Acid SCHEMBL8959846 0.81 HTR2A (0.46) ICMTHTR2AHTR2CCYP1A2CYP3A4
Fumaric Acid SCHEMBL8959840 0.81 HTR2A (0.46) ICMTHTR2AHTR2CCYP1A2CYP3A4
Fumaric Acid SCHEMBL27359202 0.81 HTR2A (0.46) ICMTHTR2AHTR2CCYP1A2CYP3A4
SCHEMBL8959663 0.78 ICMT (0.48) ICMTKCNH2
SCHEMBL8959653 0.78 ICMT (0.48) ICMTKCNH2
SCHEMBL8959664 0.73 ICMT (0.40) ICMTHTR2AHTR2CKCNH2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
CN-1105988-A 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 CN disclosed