SCHEMBL8959653

SCHEMBL8959653

CCc1cn(C[C@@H](C)O)c2ccc(F)cc12

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ICMT O60725 7/20 0.48
SCN9A Q15858 1/20 0.45
KCNH2 Q12809 1/20 0.43
CRY2 Q49AN0 9/20 0.42
PER2 O15055 8/20 0.42
CRY1 Q16526 6/20 0.42
HTR3A P46098 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8959663 1.00 ICMT (0.48) ICMTSCN9AKCNH2CRY2PER2
SCHEMBL9234058 0.86 HTR2C (0.54) ICMTKCNH2
SCHEMBL8959518 0.82 PER2 (0.40) ICMTSCN9ACRY2PER2CRY1
SCHEMBL8959520 0.82 PER2 (0.40) ICMTSCN9ACRY2PER2CRY1
Fumaric Acid SCHEMBL27342763 0.80 ICMT (0.48) ICMTHTR3A
SCHEMBL8959510 0.78 ICMT (0.45) ICMTKCNH2
SCHEMBL8959513 0.78 ICMT (0.45) ICMTKCNH2
SCHEMBL22647112 0.76 KCNH2 (0.47) ICMTKCNH2CRY2PER2CRY1
SCHEMBL13131357 0.74 ICMT (0.60) ICMTKCNH2
SCHEMBL18508879 0.73 KDM4E (0.58) ICMTKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
CN-1105988-A 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 CN disclosed
EP-0655440-A2 1-Aminoethylindoles F. HOFFMANN-LA ROCHE AG (CH) 1995-05-31 EP disclosed