SCHEMBL8959566

SCHEMBL8959566

CCc1c(C(=O)O)[nH]c2ccc(F)c(Cl)c12

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRNP P04156 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
PPARG P37231 1/20 0.48
HIF1A Q16665 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
NR2E3 Q9Y5X4 1/20 0.48
NCOR2 Q9Y618 1/20 0.48
GPR17 Q13304 4/20 0.46
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31332568 0.82 MAP2 (0.41) GPR17
SCHEMBL19331084 0.81 MEN1 (0.41) GPR17
SCHEMBL6594503 0.81 MAPT (0.47) PRNPCYP1A2CYP2C9CYP2C19PPARG
SCHEMBL31332483 0.80 MAP2 (0.43) GPR17
SCHEMBL9228790 0.80 SIRT1 (0.35) PRNPCYP1A2CYP2C9CYP2C19PPARG
SCHEMBL27397857 0.79 DAO (0.42) GPR17
SCHEMBL23000272 0.77 PRNP (0.55) PRNPCYP1A2CYP2C9CYP2C19PPARG
SCHEMBL4916175 0.74 KDM4E (0.50) CYP1A2CYP2C19MAPT
SCHEMBL266498 0.74 GPR17 (0.70) CYP1A2CYP2C9CYP2C19GPR17
SCHEMBL2538695 0.74 PRNP (0.69) PRNPCYP1A2CYP2C9CYP2C19PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
CN-1105988-A 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 CN disclosed
EP-0655440-A2 1-Aminoethylindoles F. HOFFMANN-LA ROCHE AG (CH) 1995-05-31 EP disclosed