SCHEMBL8959816

SCHEMBL8959816

OC1(c2ccc(F)cc2)C=CC=NC1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.33
HSD11B1 P28845 2/20 0.33
MAOA P21397 1/20 0.33
GRIN2B Q13224 3/20 0.33
POLB P06746 1/20 0.33
NPY5R Q15761 3/20 0.32
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CHRNA1 P02708 1/20 0.31
CHRNG P07510 1/20 0.31
CHRNB1 P11230 1/20 0.31
CHRNB2 P17787 1/20 0.31
SLC6A2 P23975 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28917498 0.83 MAOB (0.31) MAOBMAOAGRIN2BNPY5RCYP1A2
SCHEMBL29139323 0.65
SCHEMBL28308797 0.64
SCHEMBL29385800 0.63 SLC6A3 (0.37) MAOBHSD11B1MAOAMEN1KMT2A
SCHEMBL7824744 0.62 OPRM1 (0.53) MAOBMAOAPOLBSLC6A2DRD2
SCHEMBL16053689 0.61 MAOB (0.35) MAOBMAOANPY5RSLC6A3
SCHEMBL3282333 0.60
SCHEMBL7041041 0.60
SCHEMBL4800047 0.60
SCHEMBL30927080 0.59

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691956-A1 3-PHENYL-1,2,5,6-TETRAHYDROPYRIDINE DERIVATIVES AS SEDATIVES LABORATOIRE L. LAFON (FR) 1996-01-17 EP disclosed
WO-1994022827-A1 3-PHENYL-1,2,5,6-TETRAHYDROPYRIDINE DERIVATIVES AS SEDATIVES LABORATOIRE L. LAFON (FR) 1994-10-13 WO disclosed