SCHEMBL8960196

SCHEMBL8960196

CC(C)CC(SC(CC(C)C)c1ccc(Br)cc1)c1ccc(Br)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.38
MAOA P21397 1/20 0.37
PYCR1 P32322 1/20 0.37
HTR2A P28223 1/20 0.35
FPR2 P25090 1/20 0.35
CYP1A2 P05177 2/20 0.34
ALOX5 P09917 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CTSL P07711 2/20 0.34
CTSB P07858 2/20 0.34
CTSS P25774 2/20 0.34
CYP2A6 P11509 1/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP3 P08254 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9669321 0.78 CYP1A2 (0.40) MAOAPYCR1HTR2ACYP1A2ALDH1A1
SCHEMBL11389632 0.78 TAAR1 (0.42) HTR2AALDH1A1CYP3A4HSD17B10
SCHEMBL28721293 0.77 IDO1 (0.41) MAOAALDH1A1
SCHEMBL1988560 0.74 HTR2A (0.38) HTR2ACYP1A2ALDH1A1CYP3A4CYP2D6
SCHEMBL16546600 0.72 CTSK (0.38) CTSKMAOAPYCR1HTR2AFPR2
SCHEMBL11901019 0.72 CTSK (0.41) CTSKPYCR1FPR2CYP1A2ALOX5
SCHEMBL1765182 0.71 GCG (0.47) CTSKFPR2ALDH1A1CTSLCTSB
SCHEMBL28541578 0.69 ALDH1A1 (0.46) CYP1A2ALDH1A1CYP3A4HPGD
SCHEMBL24849598 0.68 SLC6A2 (0.37) PYCR1CYP1A2ALDH1A1HSD17B10
SCHEMBL16424587 0.68 CTSK (0.41) CTSKPYCR1FPR2CYP1A2ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516904-A SKIN AND IMMUNE DISORDERS; ANTIARTHRITIC AGENTS; WOUND HEALING AGENTS ALLERGAN, INC. (US) 1996-05-14 US disclosed
EP-0436398-B1 Acetylenes disubstituted with a heteroaromatic group and a substituted phenyl group having retinoid like activity ALLERGAN INC (US) 1996-01-31 EP disclosed
US-5414007-A Skin disorders ALLERGAN, INC. (US) 1995-05-09 US disclosed
US-5349105-A Skin disorder ALLERGAN, INC. (US) 1994-09-20 US disclosed
US-5264456-A Skin disorders, anticarcinogenic agents, antiarthritic agents, immunology or wound healing agents ALLERGAN, INC. (US) 1993-11-23 US disclosed
US-5202471-A Skin disorders ALLERGAN, INC. (US) 1993-04-13 US disclosed
US-5175185-A Antiacne agents ALLERGAN, INC. (US) 1992-12-29 US disclosed
EP-0436398-A1 Acetylenes disubstituted with a heteroaromatic group and a substituted phenyl group having retinoid like activity ALLERGAN, INC. (US) 1991-07-10 EP disclosed
US-5013744-A Skin disorders ALLERGAN, INC. (US) 1991-05-07 US disclosed