SCHEMBL8961670

SCHEMBL8961670

COc1cc(C(=O)N2CCC(=O)N(CC(=O)NCC(N)=O)c3ccccc32)ccc1NC(=O)c1ccccc1-c1ccc(C)cc1C

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 7/20 0.45
AVPR1B P47901 4/20 0.45
AVPR2 P30518 7/20 0.41
TP53 P04637 4/20 0.39
LMNA P02545 2/20 0.39
ALDH1A1 P00352 2/20 0.38
POLB P06746 2/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
THRB P10828 1/20 0.38
MAPT P10636 3/20 0.38
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969281 0.90 AVPR1A (0.51) AVPR1AAVPR1BAVPR2TP53LMNA
SCHEMBL6970232 0.88 AVPR1A (0.47) AVPR1AAVPR1BAVPR2TP53LMNA
SCHEMBL9414294 0.86 AVPR1A (0.47) AVPR1AAVPR1BAVPR2TP53LMNA
SCHEMBL8961732 0.84 AVPR1A (0.47) AVPR1AAVPR1BAVPR2TP53LMNA
SCHEMBL6960071 0.84 AVPR1A (0.53) AVPR1AAVPR1BAVPR2ALDH1A1PDCD1
SCHEMBL6960321 0.84 AVPR1A (0.52) AVPR1AAVPR1BAVPR2TP53LMNA
SCHEMBL6967087 0.83 AVPR1A (0.47) AVPR1AAVPR1BAVPR2TP53LMNA
SCHEMBL6970362 0.82 AVPR1A (0.49) AVPR1AAVPR1BAVPR2ALDH1A1MAPT
SCHEMBL6970821 0.81 AVPR1A (0.57) AVPR1AAVPR1BAVPR2PDCD1CD274
SCHEMBL6957577 0.80 AVPR1A (0.49) AVPR1AAVPR1BAVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5521170-A VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-28 US disclosed
EP-0620216-A1 Benzamide derivatives and their use as vasopressin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed