SCHEMBL8962836

SCHEMBL8962836

Fc1cc(-c2ccc(C3CCC(/C=C/Cl)CC3)cc2)ccc1Cl

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.35
HDAC2 Q92769 1/20 0.33
CYP11B1 P15538 4/20 0.32
CYP11B2 P19099 4/20 0.32
DGAT1 O75907 2/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
FFAR1 O14842 1/20 0.31
TRPV1 Q8NER1 1/20 0.30
DHODH Q02127 1/20 0.30
SIRT1 Q96EB6 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8962842 1.00 JAK2 (0.35) JAK2HDAC2CYP11B1CYP11B2DGAT1
SCHEMBL8963228 0.89 P2RY14 (0.35) HDAC2CYP11B1CYP11B2DGAT1NPC1
SCHEMBL8963237 0.89 P2RY14 (0.35) HDAC2CYP11B1CYP11B2DGAT1NPC1
SCHEMBL8962613 0.88 SLC6A2 (0.35) HDAC2KCNH2
SCHEMBL8962617 0.88 SLC6A2 (0.35) HDAC2KCNH2
SCHEMBL8380316 0.88 FFAR1 (0.33) JAK2HDAC2CYP11B1CYP11B2DGAT1
SCHEMBL9313856 0.88 FFAR1 (0.33) JAK2HDAC2CYP11B1CYP11B2DGAT1
SCHEMBL9313850 0.88 FFAR1 (0.33) JAK2HDAC2CYP11B1CYP11B2DGAT1
SCHEMBL8380314 0.88 FFAR1 (0.33) JAK2HDAC2CYP11B1CYP11B2DGAT1
SCHEMBL8962932 0.85 KDM1A (0.37) HDAC2NPC1RAB9AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
EP-0559860-A1 HALOVINYL-DERIVATIVES. HOFFMANN LA ROCHE (CH) 1993-09-15 EP disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed