SCHEMBL8963237

SCHEMBL8963237

Fc1ccc(-c2ccc([C@H]3CC[C@H](/C=C/Cl)CC3)cc2)cc1F

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RY14 Q15391 1/20 0.35
HDAC2 Q92769 1/20 0.34
KDM1A O60341 2/20 0.33
CYP17A1 P05093 2/20 0.33
CYP11B2 P19099 2/20 0.33
CYP3A4 P08684 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
CYP11B1 P15538 1/20 0.33
PGR P06401 3/20 0.31
KDM4E B2RXH2 1/20 0.31
CCR2 P41597 1/20 0.31
MAOB P27338 1/20 0.31
DGAT1 O75907 1/20 0.31
TNKS O95271 2/20 0.30
TNKS2 Q9H2K2 2/20 0.30
GRIN2B Q13224 1/20 0.30
SCD5 Q86SK9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963228 1.00 P2RY14 (0.35) P2RY14HDAC2KDM1ACYP17A1CYP11B2
Biphenyl SCHEMBL9450901 0.95 NPC1 (0.41) P2RY14HDAC2KDM1ACYP17A1CYP11B2
SCHEMBL8962836 0.89 JAK2 (0.35) HDAC2CYP11B2NPC1RAB9ACYP11B1
SCHEMBL8962842 0.89 JAK2 (0.35) HDAC2CYP11B2NPC1RAB9ACYP11B1
SCHEMBL9479282 0.88 HDAC2 (0.35) P2RY14HDAC2KDM1ACYP17A1CYP11B2
SCHEMBL9479289 0.88 HDAC2 (0.35) P2RY14HDAC2KDM1ACYP17A1CYP11B2
SCHEMBL9479286 0.88 HDAC2 (0.35) P2RY14HDAC2KDM1ACYP17A1CYP11B2
SCHEMBL8962808 0.88 KDM1A (0.36) HDAC2KDM1AMAOBSCD5
SCHEMBL8962817 0.88 KDM1A (0.36) HDAC2KDM1AMAOBSCD5
SCHEMBL8962846 0.87 SLC6A3 (0.39) HDAC2CYP3A4NPC1RAB9ATNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed