SCHEMBL8962916

SCHEMBL8962916

Fc1ccc(C2CCC([C@H]3CC[C@H](/C=C/Cl)CC3)CC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 1/20 0.37
DRD2 P14416 4/20 0.33
HTR1A P08908 3/20 0.33
HTR2A P28223 3/20 0.33
DRD3 P35462 3/20 0.33
DRD1 P21728 1/20 0.33
DRD5 P21918 1/20 0.33
MAP1LC3B Q9GZQ8 1/20 0.33
MAOA P21397 2/20 0.32
MAOB P27338 2/20 0.32
ESR2 Q92731 2/20 0.32
ESR1 P03372 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
KDM1A O60341 2/20 0.32
HTR2C P28335 1/20 0.31
ACHE P22303 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963034 0.89 DRD2 (0.43) HDAC2DRD2HTR1AHTR2ADRD3
SCHEMBL8963241 0.86 ESR2 (0.41) HDAC2DRD2HTR1AHTR2ADRD3
SCHEMBL9300385 0.86 ESR2 (0.41) HDAC2DRD2HTR1AHTR2ADRD3
SCHEMBL8963014 0.86 HDAC2 (0.45) HDAC2MAOAMAOBESR2ESR1
SCHEMBL8963019 0.86 HDAC2 (0.45) HDAC2MAOAMAOBESR2ESR1
SCHEMBL8963054 0.85 SLC18A3 (0.40) HDAC2DRD2CYP2C9
SCHEMBL9507875 0.85 HDAC2 (0.38) HDAC2DRD2HTR1AHTR2ADRD3
SCHEMBL9507865 0.85 HDAC2 (0.38) HDAC2DRD2HTR1AHTR2ADRD3
SCHEMBL9507869 0.85 HDAC2 (0.38) HDAC2DRD2HTR1AHTR2ADRD3
SCHEMBL9540801 0.84 DRD2 (0.40) HDAC2DRD2HTR1AHTR2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
EP-0559860-A1 HALOVINYL-DERIVATIVES. HOFFMANN LA ROCHE (CH) 1993-09-15 EP disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed