SCHEMBL8962990

SCHEMBL8962990

CCOc1ccc(-c2ccc([C@H]3CC[C@H](/C=C/Cl)CC3)cc2)cc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.44
NAAA Q02083 2/20 0.39
JAK2 O60674 1/20 0.35
NR1H4 Q96RI1 2/20 0.34
PRMT5 O14744 1/20 0.34
PTGS2 P35354 2/20 0.34
FAAH O00519 1/20 0.33
FPR2 P25090 1/20 0.33
PTGS1 P23219 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
FFAR1 O14842 1/20 0.32
PPARD Q03181 1/20 0.32
KCNQ3 O43525 1/20 0.32
KCNQ2 O43526 1/20 0.32
TUBB1 Q9H4B7 1/20 0.32
CSF1R P07333 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8962982 1.00 KDM1A (0.44) KDM1ANAAAJAK2NR1H4PRMT5
SCHEMBL8962940 0.91 HRH3 (0.36) KDM1AJAK2NR1H4PRMT5FPR2
SCHEMBL8962946 0.91 HRH3 (0.36) KDM1AJAK2NR1H4PRMT5FPR2
SCHEMBL20803726 0.91 KDM1A (0.46) KDM1ANAAANR1H4PTGS2FAAH
SCHEMBL20803723 0.89 KDM1A (0.45) KDM1ANAAANR1H4PTGS2FAAH
SCHEMBL8962824 0.87 KDM1A (0.41) KDM1ANAAAFAAH
SCHEMBL8962831 0.87 KDM1A (0.41) KDM1ANAAAFAAH
SCHEMBL20803595 0.86 KDM1A (0.46) KDM1ANAAANR1H4PTGS2FAAH
SCHEMBL20803586 0.86 KDM1A (0.46) KDM1ANAAANR1H4PTGS2FAAH
SCHEMBL22161983 0.86 KDM1A (0.46) KDM1ANAAANR1H4PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed