SCHEMBL8962831

SCHEMBL8962831

COc1ccc(-c2ccc([C@H]3CC[C@H](/C=C/Cl)CC3)cc2)cc1F

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.41
CYP17A1 P05093 1/20 0.40
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
TDP2 O95551 1/20 0.39
NAAA Q02083 8/20 0.39
ERN1 O75460 1/20 0.39
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
TGFBR1 P36897 1/20 0.36
ACVR1 Q04771 1/20 0.36
PLAT P00750 1/20 0.36
ROCK2 O75116 1/20 0.36
SCD O00767 1/20 0.36
FAAH O00519 1/20 0.35
MIF P14174 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8962824 1.00 KDM1A (0.41) KDM1ACYP17A1PDGFRBPDGFRATDP2
SCHEMBL8962990 0.87 KDM1A (0.44) KDM1ANAAAFAAH
SCHEMBL8962982 0.87 KDM1A (0.44) KDM1ANAAAFAAH
SCHEMBL8963104 0.85 JAK2 (0.34)
SCHEMBL8963112 0.85 JAK2 (0.34)
SCHEMBL8963179 0.85 CTSK (0.37) NAAAGRIN2BFAAH
SCHEMBL8963176 0.85 CTSK (0.37) NAAAGRIN2BFAAH
SCHEMBL8962940 0.85 HRH3 (0.36) KDM1A
SCHEMBL8962946 0.85 HRH3 (0.36) KDM1A
SCHEMBL20803588 0.85 KDM1A (0.43) KDM1ACYP17A1PDGFRBPDGFRATDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed