SCHEMBL8963290

SCHEMBL8963290

Clc1ccc(C2CCC([C@H]3CC[C@H](/C=C/Br)CC3)CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.41
SLC18A3 Q16572 1/20 0.39
HTR3A P46098 1/20 0.39
LSS P48449 1/20 0.37
HDAC2 Q92769 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
SLC2A1 P11166 1/20 0.36
MAPT P10636 2/20 0.35
USP2 O75604 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HIF1A Q16665 1/20 0.35
MAOA P21397 2/20 0.35
MAOB P27338 2/20 0.35
IDO1 P14902 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963054 0.85 SLC18A3 (0.40) DRD2SLC18A3HTR3ALSSHDAC2
SCHEMBL8962891 0.85 HDAC2 (0.41) SLC18A3HDAC2CYP2C9MAOAMAOB
SCHEMBL9179061 0.83 DRD2 (0.41) DRD2SLC18A3HTR3ALSSHDAC2
SCHEMBL9617265 0.83 DRD2 (0.41) DRD2SLC18A3HTR3ALSSHDAC2
SCHEMBL8962682 0.83 SLC18A3 (0.39) DRD2SLC18A3HDAC2MAPTLMNA
SCHEMBL9179048 0.83 DRD2 (0.41) DRD2SLC18A3HTR3ALSSHDAC2
SCHEMBL9300674 0.83 HDAC2 (0.37) DRD2HDAC2CYP2C9MAOAMAOB
SCHEMBL9617266 0.83 DRD2 (0.41) DRD2SLC18A3HTR3ALSSHDAC2
SCHEMBL9179054 0.83 DRD2 (0.41) DRD2SLC18A3HTR3ALSSHDAC2
SCHEMBL13557301 0.83 DRD2 (0.41) DRD2SLC18A3HTR3ALSSHDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed